Discovery of a novel potent cytochrome P450 CYP4Z1 inhibitor
David Machalz, Hongjie Li, Wei Du, Shishir Sharma, Sijie Liu, Matthias Bureik, Gerhard Wolber
Topics & Concepts
PharmacophoreChemistryIn silicoVirtual screeningDrug discoveryComputational biologyCytochrome P450EnzymeIC50BiochemistryCombinatorial chemistryIn vitroGeneBiologyPharmacogenetics and Drug MetabolismReceptor Mechanisms and SignalingComputational Drug Discovery Methods