Design, synthesis and biological evaluation of Schiff’s base derivatives as multifunctional agents for the treatment of Alzheimer’s disease
Jian Shi, Yi Zhou, Keren Wang, Qinge Ma, Rongrui Wei, Qingfeng Li, Yiyang Zhao, Zhanpin Qiao, Shuang Liu, Yumin Leng, Wenmin Liu, Zhipei Sang
Topics & Concepts
ChemistryMonoamine oxidaseSchiff baseCombinatorial chemistryLead compoundChelationIC50NeuroprotectionAntioxidantDocking (animal)Drug discoveryPharmacologyIn vitroBiochemistryStereochemistryEnzymeOrganic chemistryMedicineNursingCholinesterase and Neurodegenerative DiseasesAlzheimer's disease research and treatmentsComputational Drug Discovery Methods