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Selective and brain-penetrant lanosterol synthase inhibitors target glioma stem-like cells by inducing 24(S),25-epoxycholesterol production

Thu P. Nguyen, Wentian Wang, Alex Sternisha, Chase D. Corley, Hua-Yu Leo Wang, Xiaoyu Wang, Francisco Ortiz, Sang‐Kyun Lim, Kalil G. Abdullah, Luis F. Parada, Noelle S. Williams, Samuel K. McBrayer, Jeffrey G. McDonald, Jef K. De Brabander, Deepak Nijhawan

2023Cell chemical biology18 citationsDOIOpen Access PDF

Topics & Concepts

LanosterolPenetrant (biochemical)GliomaChemistryPharmacologySterolEnzymeBiochemistryCancer researchStereochemistryBiologyCholesterolOrganic chemistryCholesterol and Lipid MetabolismSphingolipid Metabolism and SignalingCancer, Lipids, and Metabolism
Selective and brain-penetrant lanosterol synthase inhibitors target glioma stem-like cells by inducing 24(S),25-epoxycholesterol production | Litcius