Selective and brain-penetrant lanosterol synthase inhibitors target glioma stem-like cells by inducing 24(S),25-epoxycholesterol production
Thu P. Nguyen, Wentian Wang, Alex Sternisha, Chase D. Corley, Hua-Yu Leo Wang, Xiaoyu Wang, Francisco Ortiz, Sang‐Kyun Lim, Kalil G. Abdullah, Luis F. Parada, Noelle S. Williams, Samuel K. McBrayer, Jeffrey G. McDonald, Jef K. De Brabander, Deepak Nijhawan
Topics & Concepts
LanosterolPenetrant (biochemical)GliomaChemistryPharmacologySterolEnzymeBiochemistryCancer researchStereochemistryBiologyCholesterolOrganic chemistryCholesterol and Lipid MetabolismSphingolipid Metabolism and SignalingCancer, Lipids, and Metabolism