Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP: A novel tool to probe GLP-1R pharmacology
Francis S. Willard, Joseph D. Ho, Kyle W. Sloop
Topics & Concepts
Allosteric regulationAllosteric modulatorPharmacologyMolecular PharmacologyReceptorChemistryIn vivoBiophysicsBiochemistryBiologyBiotechnologyDiabetes Treatment and ManagementReceptor Mechanisms and SignalingNeuropeptides and Animal Physiology