Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation
Neha Upadhyay, Kalpana Tilekar, Niklas Jänsch, Markus Schweipert, Jessica D. Hess, Lorena Garcia-Foncillas Macias, Piotr Mrówka, Renato J. Aguilera, Jun‐yong Choe, Franz‐Josef Meyer‐Almes, C. S. Ramaa
Topics & Concepts
ChemistryCytotoxic T cellEpigeneticsIn vitroHDAC8Cancer cellBiochemistryCancerBiologyGeneticsHistone methyltransferaseGeneHistone Deacetylase Inhibitors ResearchCholinesterase and Neurodegenerative DiseasesClick Chemistry and Applications