Next-generation epigenetic inhibitors
P. Filippakopoulos, Stefan Knapp
Abstract
Selective bromodomain inhibitors provide new opportunities to modulate transcription
Topics & Concepts
BromodomainEpigeneticsComputational biologyTranscription (linguistics)Transcription factorBiologyGeneticsGeneLinguisticsPhilosophyProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchMultiple Myeloma Research and Treatments