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Electrocatalytic multicomponent one‐pot approach to tetrahydro‐2′<i>H</i>,<scp>4<i>H</i></scp>‐spiro[benzofuran‐2,5′‐pyrimidine] scaffold

Michaïl N. Elinson, Yuliya E. Ryzhkova, A. N. Vereshchagin, Fedor V. Ryzhkov, Mikhail P. Egorov

2021Journal of Heterocyclic Chemistry11 citationsDOI

Abstract

Abstract The new electrocatalytic multicomponent transformation has been found: the electrolysis of arylaldehydes, N , N ′‐dimethylbarbiturate, and cycloxehane‐1,3‐diones in alcohols in the presence of sodium bromide as a mediator in an undivided cell results in the formation of substituted unsymmetric spirobarbituric dihydrofurans in 62%–76% yields. The optimized reaction conditions and a mechanistic rationale for this electrocatalytic multicomponent transformation are presented. This new electrocatalytic process is a facile and efficient way to produce substituted unsymmetric spirobarbituric dihydrofurans containing both barbituric and 3,5,6,7‐tetrahydro‐1‐benzofuran‐4(2 H )‐one fragments, which are promising compounds for different biomedical applications, among them are anticonvulsants, anti‐AIDS agents, and antiinflammatory remedies. The scaffold approach was employed to find a protein, which may be influenced by the synthesized compounds—human aldose reductase was proposed. It was shown by molecular docking studies that such a scaffold search is beneficial and tetrahydro‐2′ H ,4 H ‐spiro[benzofuran‐2,5′‐pyrimidines] used in this approach are promising for the development of novel aldose reductase inhibitors.

Topics & Concepts

ChemistryBenzofuranAldose reductaseCombinatorial chemistryPyrimidineSodium bromideScaffoldStereochemistryOrganic chemistrySodiumEnzymeBiomedical engineeringMedicineSulfur-Based Synthesis TechniquesRadical Photochemical ReactionsCatalytic C–H Functionalization Methods