Discovery of a potent Gilteritinib-based FLT3-PROTAC degrader for the treatment of Acute myeloid leukemia
Lei Ye, Zhenzhen Cui, Yu Sun, Haikun Zhou, Quanjin Rong, Dan Wang, Jiaming Jin, Qijian Zhang, Di Kang, Lihong Hu, Junwei Wang, Junwei Wang
Topics & Concepts
ChemistryMyeloid leukemiaCancer researchLeukemiaImmunologyMedicineProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsUbiquitin and proteasome pathways