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KRAS Mutation-Responsive miR-139-5p inhibits Colorectal Cancer Progression and is repressed by Wnt Signaling

Feng Du, Tianyu Cao, Huahong Xie, Ting Li, Lina Sun, Hao Liu, Hao Guo, Xin Wang, Qi Liu, Tae‐Wan Kim, Jeffrey L. Franklin, Ramona Graves‐Deal, Weili Han, Zuhong Tian, Minghui Ge, Yongzhan Nie, Daiming Fan, Robert J. Coffey, Yuanyuan Lu, Xiaodi Zhao

2020Theranostics63 citationsDOIOpen Access PDF

Abstract

We identified miR-139-5p as a KRAS-responsive miRNA and demonstrated its involvement in CRC progression. KRAS mutation disrupted the miR-139-5p/Wnt signaling reciprocal negative feedback mechanism, which might cause miR-139-5p downregulation and derepression of oncogenic signaling pathways and EMT. These results reveal a transcriptional regulatory mode of KRAS-driven malignant transformation and highlight miR-139-5p as a novel regulator of crosstalk between the Ras and Wnt signaling pathways in CRC.

Topics & Concepts

KRASColorectal cancerWnt signaling pathwaymicroRNACancer researchMutationMetastasisTumor progressionCancerMouse model of colorectal and intestinal cancerBiologyMedicineSignal transductionOncologyInternal medicineGeneGeneticsMicroRNA in disease regulationCancer-related molecular mechanisms researchWnt/β-catenin signaling in development and cancer
KRAS Mutation-Responsive miR-139-5p inhibits Colorectal Cancer Progression and is repressed by Wnt Signaling | Litcius