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Trends in kinase drug discovery: targets, indications and inhibitor design

Misty M. Attwood, Doriano Fabbro, Aleksandr V. Sokolov, Stefan Knapp, Helgi B. Schiöth

2021Nature Reviews Drug Discovery780 citationsDOI

Topics & Concepts

KinomeKinaseMedicineDrug discoveryClinical trialPharmacologyDrug developmentDrugImatinibAnticancer drugBioinformaticsCancer researchInternal medicineBiologyCell biologyMyeloid leukemiaChronic Myeloid Leukemia TreatmentsChronic Lymphocytic Leukemia ResearchQuinazolinone synthesis and applications
Trends in kinase drug discovery: targets, indications and inhibitor design | Litcius