RSK inhibitors as potential anticancer agents: Discovery, optimization, and challenges
Ying Sun, Lichao Tang, Chengyong Wu, Jiaxing Wang, Chengdi Wang, Chengdi Wang
Topics & Concepts
ChemistryKinaseEffectorPharmacophoreProdrugSerineDrug discoveryProtein kinase domainThreonineBiochemistryComputational biologyPhosphorylationBiologyMutantGeneMelanoma and MAPK PathwaysComputational Drug Discovery MethodsQuinazolinone synthesis and applications