Litcius/Paper detail

Design, synthesis, molecular docking and anticancer activity of benzothiazolecarbohydrazide–sulfonate conjugates: insights into ROS-induced DNA damage and tubulin polymerization inhibition

Najla Altwaijry, Mohamed A. Omar, Hanaa S. Mohamed, Marwa M. Mounier, Ahmed H. Afifi, Aladdin M. Srour

2025RSC Advances18 citationsDOIOpen Access PDF

Abstract

, respectively. Compound 6i was found to significantly elevate the ROS levels in treated cancer cells, resulting in an 8.3-fold increase in DNA fragmentation compared to untreated cells. Additionally, it raised the percentage of accumulated cells in the G2 phase from 6.85% to 18.27% in MCF-7 cells. A molecular docking technique was conducted to elucidate the binding energy, binding pose, and binding interactions of compound 6i, revealing a strong fit within the active sites of the tubulin-colchicine binding site (CBS). This study provides valuable insights into the design and synthesis of novel anticancer agents targeting tubulin polymerization.

Topics & Concepts

ConjugateBenzothiazoleChemistrySulfonatePolymerizationTubulinCombinatorial chemistryDNA damageDNADocking (animal)MicrotubuleBiophysicsStereochemistryBiochemistryOrganic chemistryPolymerBiologyCell biologySodiumMathematical analysisNursingMedicineMathematicsSynthesis and biological activitySynthesis and Biological EvaluationFerrocene Chemistry and Applications