Discovery of dioxo-benzo[b]thiophene derivatives as potent YAP-TEAD interaction inhibitors for treating breast cancer
Youngchai Son, Jaeyeal Kim, Yong‐Chan Kim, Sung-Gil Chi, Tackhoon Kim, Jinha Yu
Topics & Concepts
ChemistryDocking (animal)CTGFTranscription factorTransactivationActivator (genetics)Reporter geneCancer researchSmall moleculeStereochemistryBiochemistryGene expressionGeneGrowth factorReceptorBiologyMedicineNursingHippo pathway signaling and YAP/TAZ