Litcius/Paper detail

A widespread role for SLC transmembrane transporters in resistance to cytotoxic drugs

Enrico Girardi, Adrián César‐Razquin, Sabrina Lindinger, Κωνσταντίνος Παπακώστας, Justyna Konecka, Jennifer Hemmerich, Stefanie Kickinger, Felix Kartnig, Bettina Gürtl, Kristaps Klavins, Vitaly Sedlyarov, Álvaro Inglés‐Prieto, Giuseppe Fiume, Anna Koren, Charles-Hugues Lardeau, Richard K. Kandasamy, Stefan Kubicek, Gerhard F. Ecker, Giulio Superti‐Furga

2020Nature Chemical Biology141 citationsDOIOpen Access PDF

Topics & Concepts

TransporterOrganic cation transport proteinsBiologyATP-binding cassette transporterSolute carrier familyCytotoxic T cellDrug resistanceDrugChemical spacePharmacologyComputational biologyTransmembrane proteinDrug discoveryChemistryBiochemistryGeneticsGeneIn vitroReceptorDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesPharmacogenetics and Drug Metabolism