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Biological evaluation and molecular docking of novel 1,3,4-thiadiazole-resorcinol conjugates as multifunctional cholinesterases inhibitors

Alicja Skrzypek, Joanna Matysiak, Monika Karpińska, Kamila Czarnecka, Paweł Kręcisz, Dorota Stary, Jędrzej Kukułowicz, Beata Paw, Marek Bajda, Paweł Szymański, Andrzej Niewiadomy

2021Bioorganic Chemistry32 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryDocking (animal)StereochemistryMolecular modelAmine gas treatingEnzymeCytotoxicityCombinatorial chemistryIn vitroOrganic chemistryBiochemistryNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsPesticide Exposure and Toxicity
Biological evaluation and molecular docking of novel 1,3,4-thiadiazole-resorcinol conjugates as multifunctional cholinesterases inhibitors | Litcius