Design, synthesis, and structure−activity relationship studies of triazolo-pyrimidine derivatives as WRN inhibitors for the treatment of MSI tumors
Qibang Sui, Yuanyang Zhou, Manjia Li, Dan Wang, Rongrong Cui, Xiaoying Cai, Jia‐Bao Liu, Xiaofeng Wang, Dan Teng, Jingyi Zhou, Hui Hou, Sulin Zhang, Mingyue Zheng
Topics & Concepts
ChemistryPyrimidineStructure–activity relationshipStereochemistryPyrimidine analogueIn vitroCancer researchPharmacologyBiochemistryBiologyMedicineNeuroendocrine Tumor Research AdvancesMetastasis and carcinoma case studies