Litcius/Paper detail

Ligand binding at the protein–lipid interface: strategic considerations for drug design

Jian Payandeh, Matthew Volgraf

2021Nature Reviews Drug Discovery120 citationsDOI

Topics & Concepts

Lipid bilayerDrug discoveryPhospholipidBiophysicsSmall moleculeChemistryMembraneLigand (biochemistry)Plasma protein bindingDrugMembrane proteinBinding siteBiochemistryComputational biologyBiologyReceptorPharmacologyLipid Membrane Structure and BehaviorReceptor Mechanisms and SignalingComputational Drug Discovery Methods