Identification and characterization of isocitrate dehydrogenase 1 (IDH1) as a functional target of marine natural product grincamycin B
Zheng Wang, Zeng-xia Li, Wencao Zhao, Hongbo Huang, Jiaqi Wang, Hao Zhang, Junyan Lu, Rui-na Wang, Wei Li, Zhao Cheng, Wenlong Xu, Di Zhu, Lisha Zhou, Wei Jiang, Long Yu, Jun‐Yan Liu, Cheng Luo, Heng Zhu, Dan Ye, Weijun Pan, Jianhua Ju, Yongjun Dang
Topics & Concepts
IDH1Isocitrate dehydrogenaseBiologyGene knockdownMutantZebrafishWild typePhenotypeBiochemistryCancer researchMolecular biologyApoptosisEnzymeGeneAcute Myeloid Leukemia ResearchCancer, Hypoxia, and MetabolismProtein Degradation and Inhibitors