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3-Arylamino-quinoxaline-2-carboxamides inhibit the PI3K/Akt/mTOR signaling pathways to activate P53 and induce apoptosis

Nan‐Ying Chen, Ke Lu, Jing‐Mei Yuan, Xiaojuan Li, Zi-Yu Gu, Cheng‐Xue Pan, Dong‐Liang Mo, Gui‐Fa Su

2021Bioorganic Chemistry17 citationsDOI

Topics & Concepts

PI3K/AKT/mTOR pathwayProtein kinase BChemistryRPTORApoptosisPhosphorylationQuinoxalineSignal transductionKinaseCell biologyCell growthCancer researchBiochemistryBiologyOrganic chemistrySynthesis and Biological EvaluationQuinazolinone synthesis and applicationsSynthesis and biological activity
3-Arylamino-quinoxaline-2-carboxamides inhibit the PI3K/Akt/mTOR signaling pathways to activate P53 and induce apoptosis | Litcius