Litcius/Paper detail

A Practical Approach for the In Vitro Safety and Efficacy Assessment of an Anti-Ageing Cosmetic Cream Enriched with Functional Compounds

Nicola Zerbinati, Sabrina Sommatis, Cristina Maccario, Serena Di Francesco, Maria Chiara Capillo, Giulia Grimaldi, Raffaele Rauso, Martha Elena Mora‐Herrera, Pier Luca Bencini, Roberto Mocchi

2021Molecules15 citationsDOIOpen Access PDF

Abstract

(1) Background: Cosmeceuticals are topical products applied to human skin to prevent skin ageing and maintain a healthy skin appearance. Their effectiveness is closely linked to the compounds present in a final formulation. In this article, we propose a panel of in vitro tests to support the efficacy assessment of an anti-ageing cream enriched with functional compounds. (2) Methods: biocompatibility and the irritant effect were evaluated on reconstructed human epidermis (RHE) and corneal epithelium (HCE) 3D models. After a preliminary MTT assay, normal human dermal fibroblasts (NHDF) and keratinocytes (HaCaT) were used to evaluate the extracellular matrix (ECM) protein synthesis, and interleukin-6 (IL-6) and metalloproteinase-1 (MMP-1) production. (3) Results: data collected showed good biocompatibility and demonstrated the absence of the irritant effect in both 3D models. Therefore, we demonstrated a statistical increase in collagen and elastin productions in NHDF cells. In HaCaT cells, we highlighted an anti-inflammatory effect through a reduction in IL-6 levels in inflammatory stimulated conditions. Moreover, the reduction of MMP-1 production after UV-B radiation was demonstrated, showing significant photo-protection. (4) Conclusion: a multiple in vitro assays approach is proposed for the valid and practical assessment of the anti-ageing protection, anti-inflammatory and biocompatible claims that can be assigned to a cosmetic product containing functional compounds.

Topics & Concepts

HaCaTBiocompatibilityChemistryHuman skinIn vitroAgeingPharmacologyWound healingExtracellular matrixBiomedical engineeringMedicineBiochemistrySurgeryBiologyInternal medicineOrganic chemistryGeneticsSkin Protection and AgingBee Products Chemical AnalysisAdvancements in Transdermal Drug Delivery