Structure–activity relationship and biological evaluation of berberine derivatives as PCSK9 down-regulating agents
Tianyun Fan, Yuxin Yang, Qingxuan Zeng, Xuelei Wang, Wei Wei, Xixi Guo, Liping Zhao, Danqing Song, Yanxiang Wang, Li Wang, Bin Hong
Topics & Concepts
PCSK9KexinBerberineChemistryProprotein convertaseLDL receptorSubtilisinIn vivoPharmacologyBiochemistryLipoproteinCholesterolEnzymeBiologyBiotechnologyLipoproteins and Cardiovascular HealthBerberine and alkaloids researchMicrobial Metabolism and Applications