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Small-Molecule Compound CY-158-11 Inhibits Staphylococcus aureus Biofilm Formation

Li Shen, Jiao Zhang, Yao Chen, Lulin Rao, Xinyi Wang, Huilin Zhao, Bingjie Wang, Yanghua Xiao, Jingyi Yu, Yanlei Xu, Junhong Shi, Weihua Han, Zengqiang Song, Fangyou Yu

2023Microbiology Spectrum15 citationsDOIOpen Access PDF

Abstract

Most bacteria exist in the form of biofilms, often strongly adherent to various surfaces, causing bacterial resistance and chronic infections. In general, antibacterial drugs are not effective against biofilms. The small-molecule compound CY-158-11 inhibited the biofilm formation of S. aureus at a subinhibitory concentration. By hindering adhesion and PIA-mediated biofilm formation, CY-158-11 exhibits antibiofilm activity toward S. aureus. These findings point to a novel therapeutic agent for combating intractable S. aureus-biofilm-related infections.

Topics & Concepts

Staphylococcus aureusBiofilmMicrobiologyChemistryBiologyBacteriaGeneticsBacterial biofilms and quorum sensingAntimicrobial agents and applicationsAntimicrobial Resistance in Staphylococcus
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