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Discovery and evaluation of cytisine N-isoflavones as novel EGFR/HER2 dual inhibitors

Yanqing Wang, Xiaoying Yin, Ling‐Yan Chen, Zhixiang Yin, Zhicheng Zuo

2022Bioorganic Chemistry20 citationsDOI

Topics & Concepts

GefitinibChemistryLapatinibEpidermal growth factor receptorCytisineA431 cellsIC50PharmacologyChromoneCancer researchCancerKinaseBiochemistryCell cycleTrastuzumabCellReceptorBreast cancerBiologyMolecular medicineMedicineIn vitroStereochemistryInternal medicineNicotinic agonistHER2/EGFR in Cancer ResearchCancer therapeutics and mechanismsAdvanced Breast Cancer Therapies
Discovery and evaluation of cytisine N-isoflavones as novel EGFR/HER2 dual inhibitors | Litcius