1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
Camilla Pecoraro, Michele De Franco, Daniela Carbone, Davide Bassani, Matteo Pavan, Stella Cascioferro, Barbara Parrino, Girolamo Cirrincione, Stefano Dall’Acqua, Stefano Moro, Valentina Gandin, Patrizia Diana
Topics & Concepts
ChemistryKinaseCancer researchPancreatic cancerCancer cellApoptosisDocking (animal)EnzymeStructure–activity relationshipBiochemistryIn vivoCancerIn vitroBiologyBiotechnologyNursingMedicineGeneticsBiochemical and Molecular ResearchClick Chemistry and ApplicationsSynthesis and Characterization of Heterocyclic Compounds