Dual-target inhibitors of PARP1 in cancer therapy: A drug discovery perspective
Jiahui Zhang, Jin Zhang, Hua Li, Lixia Chen, Dahong Yao
Topics & Concepts
PARP1DruggabilityDrug discoveryPoly ADP ribose polymeraseMedicineCancerDrug developmentPharmacologyCancer researchDrugComputational biologyPolymeraseBiologyBioinformaticsEnzymeBiochemistryGeneInternal medicinePARP inhibition in cancer therapyDNA Repair MechanismsIntegrated Circuits and Semiconductor Failure Analysis