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Identification of evodiamine and rutecarpine as novel TMEM16A inhibitors and their inhibitory effects on peristalsis in isolated Guinea-pig ileum

Zhijun Zhao, Yurun Xue, Gaohua Zhang, Jie Jia, Ruilian Xiu, Yugai Jia, Yuanyuan Wang, Xiang-Chong Wang, Honglin Li, Pingping Chen, Xuan Zhang

2021European Journal of Pharmacology17 citationsDOI

Topics & Concepts

EvodiaminePeristalsisInterstitial cell of CajalInhibitory postsynaptic potentialIleumMotilityInternal medicineChemistryGuinea pigPharmacologyContraction (grammar)EndocrinologyBiologyMedicineSmooth muscleCell biologyIon Channels and ReceptorsIon Transport and Channel RegulationIon channel regulation and function
Identification of evodiamine and rutecarpine as novel TMEM16A inhibitors and their inhibitory effects on peristalsis in isolated Guinea-pig ileum | Litcius