Discovery of novel EGFR-PROTACs capable of degradation of multiple EGFR-mutated proteins
Yu Du, Shi Shi, Shu Chen, Yezi He, Wangyang Xu, Daochen Wu, Yushu Tian, Mingyang Kong, Jiahuan He, Wenhui Xie, Yijia Qiu, Yungen Xu, Yi Zou, Qihua Zhu, Qihua Zhu
Topics & Concepts
ChemistryDrug discoveryComputational biologyEGFR inhibitorsEpidermal growth factor receptorBiochemistryReceptorBiologyProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis