Discovery of highly potent and selective antiparasitic new oxadiazole and hydroxy-oxindole small molecule hybrids
Fábio S. Fernandes, Hugo Santos, Sâmia R. Lima, Caroline Conti, Manoel T. Rodrigues, Lucas A. Zeoly, Leonardo L. G. Ferreira, Renata Krogh, Adriano D. Andricopulo, Fernando Coelho
Topics & Concepts
Trypanosoma cruziBenznidazoleLeishmania infantumAntiparasiticChemistryOxindoleAntiparasitic agentChagas diseaseAmastigoteIn vitroCytotoxicityOxadiazoleStereochemistryLeishmaniaLeishmaniasisBiochemistryPharmacologyBiologyVirologyVisceral leishmaniasisOrganic chemistryImmunologyWorld Wide WebComputer scienceParasite hostingCatalysisMedicinePathologyResearch on Leishmaniasis StudiesTrypanosoma species research and implicationsSynthesis and Biological Evaluation