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Navigating the complexities of drug development for metallo-β-lactamase inhibitors

Nakita Reddy, Alessandra Moraes Balieiro, José Rogério A. Silva, Christiaan A. Gouws, Awelani Mutshembele, Per I. Arvidsson, Hendrik G. Kruger, Thavendran Govender, Tricia Naicker

2025RSC Medicinal Chemistry8 citationsDOIOpen Access PDF

Abstract

Standardized approaches to MBL inhibitor development are vital. This work highlights the benefits of uniform methodologies while addressing key preclinical challenges to bridge the gap toward successful clinical translation.

Topics & Concepts

DrugDrug developmentPharmacologyMedicineAntibiotic Resistance in BacteriaTuberculosis Research and EpidemiologyAntibiotic Use and Resistance
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