Litcius/Paper detail

hERG toxicity assessment: Useful guidelines for drug design

Amanda Garrido, Alban Lepailleur, Serge Mignani, Patrick Dallemagne, Christophe Rochais

2020European Journal of Medicinal Chemistry330 citationsDOIOpen Access PDF

Topics & Concepts

hERGPharmacologyDrugDrug developmentDrug discoveryPotassium channelCardiac toxicityChemistryComputational biologyToxicityMedicineBiologyInternal medicineBiochemistryCardiac electrophysiology and arrhythmiasIon channel regulation and functionCardiac pacing and defibrillation studies
hERG toxicity assessment: Useful guidelines for drug design | Litcius