Structural study of ponatinib in inhibiting SRC kinase
Ming Guo, Yankun Duan, Shuyan Dai, Jun Li, Xiaojuan Chen, Lingzhi Qu, Zhuchu Chen, Hudie Wei, Longying Jiang, Yongheng Chen
Topics & Concepts
PonatinibProto-oncogene tyrosine-protein kinase SrcTyrosine kinaseSH3 domainABLDasatinibKinaseProtein kinase domainMutationCancer researchBiologyCell biologyChemistryMutantBiochemistrySignal transductionGeneChronic Myeloid Leukemia TreatmentsMast cells and histamineEosinophilic Disorders and Syndromes