5-Oxohexahydroquinolines bearing 4-pyridyl methyl carboxylate as P-glycoprotein inhibitors and multidrug resistance reversal agents in cancer cells
Sara Ranjbar, Faramak Faramin Lashkarian, Mehdi Khoshneviszadeh, Fatemeh Moosavi, Amirhossein Sakhteman, Farshid Zargari, Luciano Saso, Omidreza Firuzi, Najmeh Edraki
Topics & Concepts
ChemistryP-glycoproteinMultiple drug resistanceRhodamine 123Cancer cellDoxorubicinATP-binding cassette transporterCytotoxicityPharmacologyDrug resistanceCisplatinDocking (animal)Cell cultureCytotoxic T cellEffluxBiochemistryCancerTransporterIn vitroChemotherapyAntibioticsBiologyMedicineGeneticsNursingGeneMicrobiologyDrug Transport and Resistance MechanismsMetal complexes synthesis and propertiesHIV/AIDS drug development and treatment