Litcius/Paper detail

Technologies of targeting histone deacetylase in drug discovery: Current progress and emerging prospects

Jinxiao Ru, Yuxi Wang, Zijia Li, Jiaxing Wang, Changyu Ren, Jifa Zhang

2023European Journal of Medicinal Chemistry23 citationsDOIOpen Access PDF

Topics & Concepts

Histone deacetylaseEpigeneticsChemistryHistoneDrug discoveryComputational biologySmall moleculeAcetylationPharmacologyBiochemistryBiologyGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsClick Chemistry and Applications