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Design, synthesis and biological evaluation of 1H-pyrazolo [3,4-d]pyrimidine derivatives as PAK1 inhibitors that trigger apoptosis, ER stress and anti-migration effect in MDA-MB-231 cells

Jin Zhang, Ling Zou, Pan Tang, Dabo Pan, Zhendan He, Dahong Yao

2020European Journal of Medicinal Chemistry26 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryApoptosisIC50Protein kinase BPAK1Cell growthKinaseCell biologySignal transductionCell migrationCellCancer researchBiochemistryIn vitroBiologyCell death mechanisms and regulationProtein Kinase Regulation and GTPase SignalingFOXO transcription factor regulation
Design, synthesis and biological evaluation of 1H-pyrazolo [3,4-d]pyrimidine derivatives as PAK1 inhibitors that trigger apoptosis, ER stress and anti-migration effect in MDA-MB-231 cells | Litcius