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Targeting EGFR degradation by autophagosome degraders

ZhongFeng Zhu, Jiaying Li, Shujun Shen, Hawaa Al-furas, Shengrong Li, Yichen Tong, Yi Li, Yucheng Zeng, Qianyi Feng, Kaiyue Chen, Nan Ma, Fengtao Zhou, Zhang Zhang, Zhengqiu Li, Jiyan Pang, Ke Ding, Fang Xu

2024European Journal of Medicinal Chemistry25 citationsDOIOpen Access PDF

Topics & Concepts

Epidermal growth factor receptorEGFR inhibitorsChemistryCancer researchAutophagosomeTyrosine kinaseProteolysisAutophagyReceptorBiologyBiochemistryApoptosisEnzymeProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis