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Novel smac mimetic ASTX660 (Tolinapant) and TNF-α synergistically induce necroptosis in bladder cancer cells in vitro upon apoptosis inhibition

Lei Wang, Changhua Hu, Yu Zhao, Xiaoquan Hu

2022Biochemical and Biophysical Research Communications10 citationsDOI

Topics & Concepts

NecroptosisApoptosisProgrammed cell deathTumor necrosis factor alphaCaspaseCancer cellNecrosisCell biologyBiologyCancer researchIntrinsic apoptosisCancerImmunologyBiochemistryGeneticsCell death mechanisms and regulationCancer-related Molecular PathwaysHeat shock proteins research
Novel smac mimetic ASTX660 (Tolinapant) and TNF-α synergistically induce necroptosis in bladder cancer cells in vitro upon apoptosis inhibition | Litcius