Absorption, distribution, metabolism, excretion (ADME), drug-drug interaction potential and prediction of human pharmacokinetics of SUVN-G3031, a novel histamine 3 receptor (H3R) inverse agonist in clinical development for the treatment of narcolepsy
Ramakrishna Nirogi, Gopinadh Bhyrapuneni, Nageswara Rao Muddana, Arunkumar Manoharan, Anil Shinde, Abdul Rasheed Mohammed, Nagasurya Prakash Padala, Devender Reddy Ajjala, Ramkumar Subramanian, Veera Raghava Chowdary Palacharla
Topics & Concepts
MetaboliteADMEPharmacokineticsPharmacologyChemistryInverse agonistDrug metabolismCYP3A4AgonistMetabolismCytochrome P450ReceptorBiochemistryBiologyPharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsReceptor Mechanisms and Signaling