Litcius/Paper detail

AΙ-Driven Drug Repurposing: Applications and Challenges

Paraskevi Keramida, Nikolaos Syrigos, Marousa Kouvela, Garyphallia Poulakou, Andriani Charpidou, Oraianthi Fiste

2025Medicines7 citationsDOIOpen Access PDF

Abstract

Drug repurposing is the process of discovering new therapeutic indications for already existing drugs. By using already approved molecules with known safety profiles, this approach reduces the time, costs, and failure rates associated with traditional drug development, accelerating the availability of new treatments to patients. Artificial Intelligence (AI) plays a crucial role in drug repurposing by exploiting various computational techniques to analyze and process big datasets of biological and medical information, predict similarities between biomolecules, and identify disease mechanisms. The purpose of this review is to explore the role of AI tools in drug repurposing and underline their applications across various medical domains, mainly in oncology, neurodegenerative disorders, and rare diseases. However, several challenges remain to be addressed. These include the need for a deeper understanding of molecular mechanisms, ethical concerns, regulatory requirements, and issues related to data quality and interpretability. Overall, AI-driven drug repurposing is an innovative and promising field that can transform medical research and drug development, covering unmet medical needs efficiently and cost-effectively.

Topics & Concepts

Drug repositioningRepurposingDrugDrug discoveryProcess (computing)Computer scienceRisk analysis (engineering)Drug developmentField (mathematics)Big dataData scienceMedicineMedical researchApproved drugDiseaseBenchmark (surveying)Precision medicineQuality (philosophy)PharmacologyManagement scienceComputational Drug Discovery Methodsvaccines and immunoinformatics approachesCell Image Analysis Techniques