GPCR activation and GRK2 assembly by a biased intracellular agonist
Jia Duan, Heng Liu, Fenghui Zhao, Qingning Yuan, Yujie Ji, Xiaoqing Cai, Xinheng He, Xinzhu Li, Junrui Li, Kaichun Wu, Tianyu Gao, Shengnan Zhu, Shi Lin, Ming‐Wei Wang, Xi Cheng, Wanchao Yin, Yi Jiang, Dehua Yang, H. Eric Xu
Topics & Concepts
G protein-coupled receptor kinaseG protein-coupled receptorBeta adrenergic receptor kinaseG proteinArrestinReceptorCell biologyChemistryNeurotensin receptorRhodopsin-like receptorsBiologyBiochemistryAgonistNeurotensinNeuropeptideMetabotropic receptorReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyProtein Kinase Regulation and GTPase Signaling