From lead to clinic: A review of the structural design of P2X7R antagonists
Ruijia Zhang, Na Li, Min Zhao, Minghai Tang, Xueqin Jiang, Xiaoying Cai, Neng Ye, Kaiyue Su, Jing Peng, Xinlu Zhang, Wenshuang Wu, Haoyu Ye, Haoyu Ye
Topics & Concepts
Purinergic receptorProinflammatory cytokineReceptorImmune systemDownregulation and upregulationMultiple sclerosisChemistryArthritisInflammationPharmacologyNeuroscienceImmunologyMedicineBiologyBiochemistryGeneAdenosine and Purinergic SignalingMast cells and histamineN-Heterocyclic Carbenes in Organic and Inorganic Chemistry