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Biocatalytic access to betazole using a one-pot multienzymatic system in continuous flow

María Romero‐Fernández, Francesca Paradisi

2021Green Chemistry39 citationsDOIOpen Access PDF

Abstract

The primary amine of betazole is synthesised from an alcohol in a one-pot, continuous flow biocatalytic cascade, using a PBR hosting a multienzyme co-immobilised system with constant O<sub>2</sub> supply for <italic>in situ</italic> cofactor recycling, yielding 2.59 g L<sup>−1</sup> h<sup>−1</sup>.

Topics & Concepts

Amine gas treatingChemistryContinuous flowAlcoholCascadePrimary alcoholPrimary (astronomy)Organic chemistryFlow chemistryCofactorCombinatorial chemistryChromatographyCatalysisEnzymePhysicsMechanicsAstronomyInnovative Microfluidic and Catalytic Techniques InnovationEnzyme Catalysis and ImmobilizationAsymmetric Hydrogenation and Catalysis
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