Multiple post-translational modifications ensure EGFR functionality: Potential therapeutic targets to overcome its drug-resistance mutations
Qiangqiang He, Meiyu Qu, Hangyang Bao, Yana Xu, Tingyu Shen, Dan Tan, Muhammad Qasim Barkat, Chengyun Xu, Linghui Zeng, Ximei Wu
Topics & Concepts
T790MCancer researchEpidermal growth factor receptorGefitinibAutophosphorylationCyclin-dependent kinase 8MutationTyrosine kinaseEGFR inhibitorsBiologyKinaseCancerSignal transductionProtein kinase AGeneticsGeneNotch signaling pathwayLung Cancer Treatments and MutationsPeptidase Inhibition and AnalysisPI3K/AKT/mTOR signaling in cancer