Bis(vinylsulfonyl)piperazines as efficient linkers for highly homogeneous antibody-drug conjugates
Rong Huang, Yao Sheng, Wei Ding, Jianghui Yu, Hongli Chen, Biao Jiang
Topics & Concepts
ChemistryConjugateCombinatorial chemistryCytotoxicityHomogeneousAntibodyStereochemistryDisulfide bondIn vitroDrugBiochemistryPsychiatryMathematicsBiologyPsychologyPhysicsImmunologyThermodynamicsMathematical analysisMonoclonal and Polyclonal Antibodies ResearchHER2/EGFR in Cancer ResearchClick Chemistry and Applications