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Design, synthesis, and pharmacological evaluation of novel benzothiazole derivatives targeting LCK in acute lymphoblastic leukemia

Yanmei Chen, Kai Zhang, Jiacheng Tan, Zhichao Fan, Yuqi Fu, Xiang Li, Bo Liu, Guan Wang

2024Bioorganic Chemistry13 citationsDOI

Topics & Concepts

ChemistryTyrosine kinaseBenzothiazoleSrc family kinaseLeukemiaCancer researchKinaseApoptosisCell growthProto-oncogene tyrosine-protein kinase SrcSignal transductionCell biologyJurkat cellsCell cycleBiochemistryT cellBiologyImmune systemImmunologyAcute Lymphoblastic Leukemia researchChronic Myeloid Leukemia TreatmentsQuinazolinone synthesis and applications
Design, synthesis, and pharmacological evaluation of novel benzothiazole derivatives targeting LCK in acute lymphoblastic leukemia | Litcius