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Oxygen Surrogate Systems for Supporting Human Drug-Metabolizing Cytochrome P450 Enzymes

Silja J. Strohmaier, James J. De Voss, Ulrik Jurva, Shalini Andersson, Elizabeth M. J. Gillam

2020Drug Metabolism and Disposition15 citationsDOIOpen Access PDF

Topics & Concepts

Cytochrome P450CYP1A2ChemistryMonooxygenaseSubstrate (aquarium)RedoxBiocatalysisEnzyme kineticsCumene hydroperoxideEnzymeHydrogen peroxideCYP3A4Combinatorial chemistryCYP2B6Drug metabolismCYP2C19BiochemistryStereochemistryActive siteCatalysisOrganic chemistryBiologyReaction mechanismEcologyPharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsCancer Treatment and Pharmacology