A NSD3-targeted PROTAC suppresses NSD3 and cMyc oncogenic nodes in cancer cells
Chenxi Xu, Fanye Meng, Kwang‐Su Park, Aaron J. Storey, Weida Gong, Yi‐Hsuan Tsai, Elisa Gibson, Stephanie D. Byrum, Dongxu Li, Rick D. Edmondson, Samuel G. Mackintosh, Masoud Vedadi, Ling Cai, Alan J. Tackett, H. Ümit Kanıskan, Jian Jin, Gang Greg Wang
Topics & Concepts
Cancer researchCRISPRCell biologyPAS domainBiologyChemistryGeneGeneticsTranscription factorProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis