Litcius/Paper detail

Interleukin-1β, Oxidative Stress, and Abnormal Calcium Handling Mediate Diabetic Arrhythmic Risk

Hong Liu, Yang Zhao, An Xie, Tae Yun Kim, Radmila Terentyeva, Man Liu, Guangbin Shi, Feng Feng, Bum‐Rak Choi, Dmitry Terentyev, Shanna Hamilton, Samuel C. Dudley

2021JACC Basic to Translational Science54 citationsDOIOpen Access PDF

Abstract

Diabetes mellitus (DM) is associated with increased arrhythmia. Type 2 DM (T2DM) mice showed prolonged QT interval and increased ventricular arrhythmic inducibility, accompanied by elevated cardiac interleukin (IL)-1β, increased mitochondrial reactive oxygen species (mitoROS), and oxidation of the sarcoplasmic reticulum (SR) Ca2+ release channel (ryanodine receptor 2 [RyR2]). Inhibiting IL-1β and mitoROS reduced RyR2 oxidation and the ventricular arrhythmia in DM. Inhibiting SR Ca2+ leak by stabilizing the oxidized RyR2 channel reversed the diabetic arrhythmic risk. In conclusion, cardiac IL-1β mediated the DM-associated arrhythmia through mitoROS generation that enhances SR Ca2+ leak. The mechanistic link between inflammation and arrhythmias provides new therapeutic options.

Topics & Concepts

Ryanodine receptor 2Ryanodine receptorOxidative stressInternal medicineMedicineDiabetes mellitusEndocrinologyCalciumReactive oxygen speciesDiabetic cardiomyopathyInflammationCardiac arrhythmiaCardiologyChemistryHeart failureAtrial fibrillationBiochemistryCardiomyopathyCardiac electrophysiology and arrhythmiasIon channel regulation and functionHeart Rate Variability and Autonomic Control