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Probing 4-(diethylamino)-salicylaldehyde-based thiosemicarbazones as multi-target directed ligands against cholinesterases, carbonic anhydrases and α-glycosidase enzymes

Sadaf Hashmi, Samra Khan, Zahid Shafiq, Parham Taslımı, Muhamamd Ishaq, Nastaran Sadeghian, Halide Sedef Karaman, Naeem Akhtar, Muhammad Islam, Asnuzilawati Asari, Habsah Mohamad, İlhami Gülçın

2020Bioorganic Chemistry86 citationsDOI

Topics & Concepts

ChemistrySalicylaldehydeEnzymeButyrylcholinesteraseGlycoside hydrolaseStereochemistryCholinesterasePyrrolineGene isoformIsozymeSemicarbazoneBiochemistryAchéAcetylcholinesterasePharmacologySchiff baseMedicineGeneCholinesterase and Neurodegenerative DiseasesEnzyme function and inhibitionPhenothiazines and Benzothiazines Synthesis and Activities
Probing 4-(diethylamino)-salicylaldehyde-based thiosemicarbazones as multi-target directed ligands against cholinesterases, carbonic anhydrases and α-glycosidase enzymes | Litcius