Litcius/Paper detail

Design, synthesis and biological evaluation of novel carbamates as potential inhibitors of acetylcholinesterase and butyrylcholinesterase

Jie Wu, Marco Pistolozzi, Siyu Liu, Wen Tan

2020Bioorganic & Medicinal Chemistry37 citationsDOIOpen Access PDF

Topics & Concepts

ButyrylcholinesteraseAcetylcholinesteraseChemistryRivastigmineCholinesteraseAchéPharmacologyIC50EnzymeStereochemistryIn vitroDonepezilBiochemistryDementiaInternal medicineDiseaseMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsMedicinal Plants and Neuroprotection