A head-to-head comparison of the inhibitory activities of 15 peptidomimetic SARS-CoV-2 3CLpro inhibitors
Subramanyam Vankadara, Yun Xuan Wong, Bo Liu, Yi Yang See, Li Tan, Qian Tan, Gang Wang, Ratna Karuna, Xue Guo, Shu Ting Tan, Jia Yi Fong, Joma Joy, C. S. Brian Chia
Topics & Concepts
PeptidomimeticChemistrySevere acute respiratory syndrome coronavirus 2 (SARS-CoV-2)PharmacologyCoronavirus disease 2019 (COVID-19)ProteaseVirologyMedicineBiochemistryEnzymeInternal medicineDiseasePeptideInfectious disease (medical specialty)SARS-CoV-2 and COVID-19 ResearchComputational Drug Discovery Methodsvaccines and immunoinformatics approaches